生物活性抑制剂报价

2017/10/19 13:30:12  作者:腾准&思域


 

生物活性抑制剂是一类具有高生物活性的特殊小分子杂环化合物,这些小分子在生物体内通过氢键、疏水作用以及色散力等与特定的抗体及酶相互作用,使相应蛋白的二级结构和三级结构发生变化,从而起到一定的蛋白抑制活性。


试剂列表

 

货号 cas号 品名/规格纯度 分子式 查询/购买
N824559 177355-84-9 DBeQ, 99%  N,N'-Dibenzyl-2,4-quinazolinediamine, 99% C22H20N4 购买
D824560 252017-04-2 4-[[3-氯-4-[[(2R)-3,3,3-三氟-2-羟基-2-甲基-1-氧代丙基]氨基]苯基]磺酰基]-N,N-二甲基苯甲酰胺, 99%  (2,4-Dihydroxy-5-isopropylphenyl)5-[(4-methyl-1-piperazinyl)meth yl]-1,3-dihydro-2H-isoindol-2-ylmethanone, 99% C19H18ClF3N2O5S 购买
G824562 1086062-66-9 2,4-二氟-n-[2-甲氧基-5-[4-(4-吡嗪)-6-喹啉]-3-吡啶]苯磺酰胺, 99%  GSK-2126458, 99% C25H17F2N5O3S 购买
P815933 82508-31-4 土槿皮乙酸, 分析对照品  Pseudolaric acid B, 分析对照品 C23H28O8 购买
D824563 912999-49-6 AT-13387, 99%  (2,4-dihydroxy-5-propan-2-ylphenyl)-[5-[(4-methylpiperazin-1-yl)methyl]-1,3-dihydroisoindol-2-yl]methanone, 99% C24H31N3O3 购买
C824564 848695-25-0 6-氯-9-((4-甲氧基-3,5-二甲基吡啶-2-基)甲基)-9H-嘌呤-2-胺, 99%  6-Chloro-9-((4-methoxy-3,5-dimethylpyridin-2-yl)methyl)-9H-purin-2-amine, 99% C14H15ClN6O 购买
N824565 1206101-20-3 N-(5-(4-((6-氰基吡啶-3-基)甲氧基)苯基)-[1,2,4]噻唑并[1,5-a]吡啶-2-基)环丙烷羧酰胺, 99%  N-[5-[4-[(6-Cyano-3-pyridinyl)methoxy]phenyl][1,2,4]triazolo[1,5-a]pyridin-2-yl] cyclopropanecarboxamide, 99% C23H18N6O2 购买
N824615 1197160-78-3 N-[4-[[4-(二甲基氨基)-1-哌啶基]羰基]苯基]-N’-[4-[4,6-二(4-吗啉基)-1,3,5-三嗪-2-基]苯基]脲, 99%  N-[4-[[4-(Dimethylamino)-1-piperidinyl]carbonyl]phenyl]-N'-[4-(4,6-di-4-morpholinyl-1,3,5-triazin-2-yl)phenyl]-urea, 99% C32H41N9O4 购买
N824566 1029712-80-8 2-氟-N-甲基-4-[7-[(喹啉-6-基)甲基]咪唑并[1,2-B]-[1,2,4]三嗪-2-基]苯甲酰胺, 99%  2-fluoro-N-methyl-4-[7-(quinolin-6-ylmethyl)imidazo[1,2-b][1,2,4]triazin-2-yl]benzamide, 99% C23H17FN6O 购买
T824567 300801-52-9 (Z)-1-(3-乙基-5-甲氧基-2,3-二羟基并噻唑-2-亚基)丙酮, 99%  TG003, 99% C13H15NO2S 购买
M824572 338967-87-6 Mdivi-1, 99%  Mdivi-1, 99% C15H10Cl2N2O2S 购买
S824573 1009298-59-2 3-[2,4-双((3S)-3-甲基吗啉-4-基)吡啶并[5,6-E]嘧啶-7-基]-N-甲基苯甲酰胺, 99%  3-[2,4-bis[(3S)-3-methylmorpholin-4-yl]pyrido[2,3-d]pyrimidin-7-yl]-N-methylbenzamide, 99% C25H30N6O3 购买
T824574 1252003-15-8 Tubastatin A, 99%  Tubastatin A, 99% C20H21N3O2 购买
K824609 1469337-95-8 K-Ras(G12C) inhibitor 12, 97%  K-Ras(G12C) inhibitor 12, 97% C15H17ClIN3O3 购买
K824608 1469337-91-4 K-Ras(G12C) inhibitor 9, 99%  K-Ras(G12C) inhibitor 9, 99% C16H21ClIN3O4S 购买
H824614 1469338-01-9 6H05, 99%  6H05, 99% C20H30ClN3O2S3.CF3COOH 购买
R823899 877399-52-5 3-[(1R)-1-(2,6-二氯-3-氟苯基)乙氧基]-5-[1-(4-哌啶)-1H-吡唑-4-基]-2-吡啶胺, 98%  3-[(1R)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-[1-(4-piperidinyl)-1H-pyrazol-4-yl]-2-Pyridinamine, 98% C21H22Cl2FN5O 购买
P824605 292605-14-2 SB-3CT, 99%  2-[(4-phenoxyphenyl)sulfonylmethyl]thiirane, 99% C15H14O3S2 购买
R824606 168273-06-1 利莫那班, 99%  Rimonabant, 99% C22H21Cl3N4O 购买
Z824607 667463-62-9 (2'Z,3'E)-6-溴靛玉红-3'-肟, 99%  (2'Z,3'E)-6-Bromoindirubin-3'-oxim, 99% C16H10BrN3O2 购买
T824603 49671-76-3 2-(4-叔丁基苯基)苯并咪唑, 98%  2-(4-tert-butylphenyl)-1h-benzo[d]imidazole, 98% C17H18N2 购买
E824600 1395084-25-9 4-[(1E)-2-(2-氨基-4-羟基-5-甲基苯基)偶氮]-N-2-吡啶基苯磺酰胺, 98%  (E)-4-((2-amino-4-hydroxy-5-methylphenyl)diazenyl)-N-(pyridin-2-yl)benzenesulfonamide, 98% C18H17N5O3S 购买
H824599 1374601-40-7 BRD4770, 98%  methyl 2-benzamido-1-(3-phenylpropyl)-1H-benzo[d]imidazole-5-carboxylate, 98% C25H23N3O3 购买
M824598 10936341-25-0 6-马来酰亚胺基己酸-N-羟基琥珀酰亚胺酯, 98%  6-Maleimidohexanoic acid N-hydroxysuccinimide ester, 98% C35H43N7O11 购买
M824597 159857-81-5 马来酰亚胺基己酰-L-缬氨酸-L-瓜氨酸对氨基苄醇对硝基苯基碳酸脂, 98%  Maleimidocaproyl-L-valine-L-citrulline-p-aminobenzyl alcohol p-nitrophenyl carbonate, 98% C35H43N7O11 购买
M824596 55750-63-5 6-(马来酰亚胺基)己酸琥珀酰亚胺酯, 98%  6-Maleimidohexanoic acid N-hydroxysuccinimide ester, 98% C14H16N2O6 购买
S824595 1260907-17-2 (4S)-6-(4-氯苯基)-N-乙基-8-甲氧基-1-甲基-4H-[1,2,4]三唑并[4,3-A][1,4]苯并二氮杂卓-4-乙酰胺, 99%  (4S)-6-(4-Chlorophenyl)-N-ethyl-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepine-4-acetamide, 99% C22H22ClN5O2 购买
D824594 183232-66-8 1-(2,4-二氯苯基)-5-(4-碘苯基)-4-甲基-N-(哌啶-1-基)-1H-吡唑-3-甲酰胺, 99%  1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-n-1-piperidinyl-1 h-pyrazole-3-carboxamide, 99% C22H21Cl2IN4O 购买
E824593 1009817-63-3 (3E,5E)-3,5-二[(4-硝基苯基)亚甲基]-1-(1-氧代-2-丙烯-1-基)-4-哌啶酮, 99%  (3E,5E)-3,5-Bis[(4-nitrophenyl)methylene]-1-(1-oxo-2-propen-1-yl)-4-piperidinone, 99% C22H17N3O6 购买
T824591 1392399-03-9 BIX 01294, 99%  Trihydrochloride Hydrate, 99% C28H38N6O2.3HCl 购买
N824589 326914-06-1 MHY1485, 98%  4,6-dimorpholino-N-(4-nitrophenyl)-1,3,5-triazin-2-amine, 98% C17H21N7O4 购买
L824616 668467-91-2 LDN-57444, 97%  LDN-57444, 97% C17H11Cl3N2O3 购买
N824585 362003-83-6 NVP-231, 98%  N-[2-(Benzoylamino)-6-benzothiazolyl]tricyclo[3.3.1.13,7]decane-1-carboxamide, 98% C25H25N3O2S 购买
R824583 162011-90-7 罗非昔布, 98%  Rofecoxib, 98% C17H14O4S 购买
A824581 486424-20-8 3-氨基-6-[4-[(4-甲基-1-哌嗪基)磺酰基]苯基]-N-3-吡啶基-吡嗪甲酰胺, 98%  AZD-2858, 98% C21H23N7O3S 购买
P824577 303727-31-3 4-(4-氯-3-羟基苯基)-2-苯基-5-(吡啶-4-基)-1H-咪唑, 98%  2-(Phenyl)-4-(3-hydroxy-4-chlorophenyl)-5-(4-pyridyl)-1H-imidazole, 98% C20H14ClN3O 购买

 

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